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Academic Journal

Colombian Contributions Fighting Leishmaniasis: A Systematic Review on Antileishmanials Combined with Chemoinformatics Analysis.

  • Authors : Sánchez-Suárez J; Bioprospecting Research Group, School of Engineering, Universidad de La Sabana, Chía 250001, Colombia.; Bernal FA

Subjects: Antiprotozoal Agents/Antiprotozoal Agents/Antiprotozoal Agents/*therapeutic use ; Leishmania/Leishmania/Leishmania/*drug effects ; Leishmaniasis, Cutaneous/Leishmaniasis, Cutaneous/Leishmaniasis, Cutaneous/*drug therapy

  • Source: Molecules (Basel, Switzerland) [Molecules] 2020 Dec 03; Vol. 25 (23). Date of Electronic Publication: 2020 Dec 03.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium:

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Academic Journal

Identification of Potential Kinase Inhibitors within the PI3K/AKT Pathway of Leishmania Species.

  • Authors : Ochoa R; Programa de Estudio y Control de Enfermedades Tropicales PECET, Faculty of Medicine, University of Antioquia, Medellín 050010, Colombia.; Biophysics of Tropical Diseases Max Planck Tandem Group, University of Antioquia, Medellín 050010, Colombia.

Subjects: Leishmania/Leishmania/Leishmania/*drug effects ; Leishmania/Leishmania/Leishmania/*metabolism ; Protein Kinase Inhibitors/Protein Kinase Inhibitors/Protein Kinase Inhibitors/*chemistry

  • Source: Biomolecules [Biomolecules] 2021 Jul 16; Vol. 11 (7). Date of Electronic Publication: 2021 Jul 16.Publisher: MDPI Country of Publication: Switzerland NLM ID: 101596414 Publication Model: Electronic Cited Medium:

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Academic Journal

Identification of Kaurane-Type Diterpenes as Inhibitors of Leishmania Pteridine Reductase I.

  • Authors : Herrera-Acevedo C; Post-Graduate Program in Natural and Synthetic Bioactive Products, Federal University of Paraíba, João Pessoa 58051-900, PB, Brazil.; Bioorganic Chemistry Laboratory, Facultad de Ciencias Básicas y Aplicadas, Universidad Militar Nueva Granada, Cajicá 250247, Colombia.

Subjects: Diterpenes, Kaurane/Diterpenes, Kaurane/Diterpenes, Kaurane/*pharmacology ; Enzyme Inhibitors/Enzyme Inhibitors/Enzyme Inhibitors/*pharmacology ; Leishmania/Leishmania/Leishmania/*enzymology

  • Source: Molecules (Basel, Switzerland) [Molecules] 2021 May 21; Vol. 26 (11). Date of Electronic Publication: 2021 May 21.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium:

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Academic Journal

Hybrid Cyclobutane/Proline-Containing Peptidomimetics: The Conformational Constraint Influences Their Cell-Penetration Ability.

  • Authors : Illa O; Departament de Química, Universitat Autònoma de Barcelona, 08193 Cerdanyola del Vallès, Spain.; Ospina J

Subjects: Cell-Penetrating Peptides/Cell-Penetrating Peptides/Cell-Penetrating Peptides/*metabolism ; Cyclobutanes/Cyclobutanes/Cyclobutanes/*metabolism ; Leishmania/Leishmania/Leishmania/*metabolism

  • Source: International journal of molecular sciences [Int J Mol Sci] 2021 May 11; Vol. 22 (10). Date of Electronic Publication: 2021 May 11.Publisher: MDPI Country of Publication: Switzerland NLM ID: 101092791 Publication Model: Electronic Cited Medium:

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Academic Journal

In Vitro Anti-Leishmanial Effect of Metallic Meso-Substituted Porphyrin Derivatives against Leishmania braziliensis and Leishmania panamensis Promastigotes Properties.

Subjects: Leishmania/Leishmania/Leishmania/*drug effects ; Leishmania braziliensis/Leishmania braziliensis/Leishmania braziliensis/*drug effects ; Metalloporphyrins/Metalloporphyrins/Metalloporphyrins/*chemistry

  • Source: Molecules (Basel, Switzerland) [Molecules] 2020 Apr 19; Vol. 25 (8). Date of Electronic Publication: 2020 Apr 19.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium:

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Academic Journal

Synthesis and Evaluation of Antileishmanial and Cytotoxic Activity of Benzothiopyrane Derivatives.

  • Authors : Ortiz C; Química Orgánica de Productos Naturales, Instituto de Química, Facultad de Ciencias Exactas y Naturales, Universidad de Antioquia, calle 70, No. 52-21, Medellín A. A 1226, Colombia.; Echeverri F

Subjects: Antiprotozoal Agents/Antiprotozoal Agents/Antiprotozoal Agents/*pharmacology ; Cell Proliferation/Cell Proliferation/Cell Proliferation/*drug effects ; Leishmania/Leishmania/Leishmania/*drug effects

  • Source: Molecules (Basel, Switzerland) [Molecules] 2020 Feb 12; Vol. 25 (4). Date of Electronic Publication: 2020 Feb 12.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium:

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Academic Journal

Synthesis and Evaluation of Thiochroman-4-One Derivatives as Potential Leishmanicidal Agents.

  • Authors : Vargas E; Química Orgánica de Productos Naturales, Instituto de Química, Facultad de Ciencias Exactas y Naturales, Universidad de Antioquia, calle 70 No. 52-21, Medellin A.A 1226, Colombia. .; Echeverri F

Subjects: Antiprotozoal Agents/Antiprotozoal Agents/Antiprotozoal Agents/*chemical synthesis ; Antiprotozoal Agents/Antiprotozoal Agents/Antiprotozoal Agents/*pharmacology ; Leishmania/Leishmania/Leishmania/*drug effects

  • Source: Molecules (Basel, Switzerland) [Molecules] 2017 Nov 29; Vol. 22 (12). Date of Electronic Publication: 2017 Nov 29.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium:

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Academic Journal

Synthesis of Novel Quaternary Ammonium Salts and Their in Vitro Antileishmanial Activity and U-937 Cell Cytotoxicity.

Subjects: Ammonium Compounds/Ammonium Compounds/Ammonium Compounds/*chemistry ; Leishmania/Leishmania/Leishmania/*drug effects ; Leishmaniasis/Leishmaniasis/Leishmaniasis/*drug therapy

  • Source: Molecules (Basel, Switzerland) [Molecules] 2016 Mar 29; Vol. 21 (4), pp. 381. Date of Electronic Publication: 2016 Mar 29.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium:

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Academic Journal

Synthesis, leishmanicidal and cytotoxic activity of triclosan-chalcone, triclosan-chromone and triclosan-coumarin hybrids.

  • Authors : Otero E; Química de Plantas Colombianas, Instituto de Química, Facultad de Ciencias Exactas y Naturales, Universidad de Antioquia UdeA, Calle 70 No. 52-21, A.A 1226 Medellín, Colombia. .; Vergara S

Subjects: Antiprotozoal Agents/Antiprotozoal Agents/Antiprotozoal Agents/*pharmacology ; Chalcones/Chalcones/Chalcones/*pharmacology ; Coumarins/Coumarins/Coumarins/*pharmacology

  • Source: Molecules (Basel, Switzerland) [Molecules] 2014 Aug 28; Vol. 19 (9), pp. 13251-66. Date of Electronic Publication: 2014 Aug 28.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium:

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Academic Journal

In-silico analyses of sesquiterpene-related compounds on selected Leishmania enzyme-based targets.

  • Authors : Bernal FA; Laboratorio de Química Bioorgánica, Departamento de Química, Facultad de Ciencias Básicas y Aplicadas, Universidad Militar Nueva Granada, Cundinamarca 250240, AA 49300, Colombia. .; Coy-Barrera E

Subjects: Drug Design*; Leishmania/Leishmania/Leishmania/*drug effects ; Leishmaniasis/Leishmaniasis/Leishmaniasis/*drug therapy

  • Source: Molecules (Basel, Switzerland) [Molecules] 2014 Apr 29; Vol. 19 (5), pp. 5550-69. Date of Electronic Publication: 2014 Apr 29.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium:

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