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Academic Journal

Molecular Docking-Based Virtual Screening of FDA-Approved Drugs Using Trypanothione Reductase Identified New Trypanocidal Agents.

  • Authors : Gómez-Escobedo R; Departamento de Parasitología, Escuela Nacional de Ciencias Biológicas, Instituto Politécnico Nacional, Ciudad de México 07738, Mexico.; Méndez-Álvarez D

Subjects: Trypanocidal Agents*/Trypanocidal Agents*/Trypanocidal Agents*/pharmacology ; Trypanocidal Agents*/Trypanocidal Agents*/Trypanocidal Agents*/chemistry ; NADH, NADPH Oxidoreductases*/NADH, NADPH Oxidoreductases*/NADH, NADPH Oxidoreductases*/antagonists & inhibitors

  • Source: Molecules (Basel, Switzerland) [Molecules] 2024 Aug 10; Vol. 29 (16). Date of Electronic Publication: 2024 Aug 10.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049

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Academic Journal

Efficacy of short-course treatment for prevention of congenital transmission of Chagas disease: A retrospective cohort study.

  • Authors : Moscatelli G; Servicio de Parasitología y Chagas, Hospital de Niños 'Ricardo Gutiérrez', Buenos Aires, Argentina.; Instituto Multidisciplinario de Investigaciones en Patologías Pediatricas (IMIPP)- CONICET-GCBA, Buenos Aires, Argentina.

Subjects: Chagas Disease*/Chagas Disease*/Chagas Disease*/drug therapy ; Chagas Disease*/Chagas Disease*/Chagas Disease*/prevention & control ; Nitroimidazoles*/Nitroimidazoles*/Nitroimidazoles*/therapeutic use

  • Source: PLoS neglected tropical diseases [PLoS Negl Trop Dis] 2024 Jan 22; Vol. 18 (1), pp. e0011895. Date of Electronic Publication: 2024 Jan 22 (Print Publication: 2024).Publisher: Public Library of Science Country of Publication: United States NLM ID: 101291488 Publication Model: eCollection Cited Medium: Internet

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Academic Journal

ELISA F29 -A therapeutic efficacy biomarker in Chagas disease: Evaluation in pediatric patients treated with nifurtimox and followed for 4 years post-treatment.

Subjects: Trypanocidal Agents*/Trypanocidal Agents*/Trypanocidal Agents*/therapeutic use ; Chagas Disease*/Chagas Disease*/Chagas Disease*/diagnosis ; Chagas Disease*/Chagas Disease*/Chagas Disease*/drug therapy

  • Source: PLoS neglected tropical diseases [PLoS Negl Trop Dis] 2023 Jun 23; Vol. 17 (6), pp. e0011440. Date of Electronic Publication: 2023 Jun 23 (Print Publication: 2023).Publisher: Public Library of Science Country of Publication: United States NLM ID: 101291488 Publication Model: eCollection Cited Medium: Internet

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Academic Journal

Population pharmacokinetics of benznidazole in neonates, infants and children using a new pediatric formulation.

  • Authors : Altcheh J; Servicio de Parasitologia y Chagas, Hospital de Niños 'Dr Ricardo Gutierrez', Buenos Aires, Argentina.; PEDCHAGAS Network (Hospital de Niños Ricardo Gutiérrez, Hospital de Niños Doctor Hector Quintana, Hospital Público Materno Infantil, Centro de Chagas y Patología Regional de Santiago del Estero, & Instituto Nacional de Parasitología Dr. Mario Fatala Chaben), Argentina.

Subjects: Chagas Disease*/Chagas Disease*/Chagas Disease*/drug therapy ; Nitroimidazoles*/Nitroimidazoles*/Nitroimidazoles*/therapeutic use ; Trypanocidal Agents*/Trypanocidal Agents*/Trypanocidal Agents*/therapeutic use

  • Source: PLoS neglected tropical diseases [PLoS Negl Trop Dis] 2023 May 31; Vol. 17 (5), pp. e0010850. Date of Electronic Publication: 2023 May 31 (Print Publication: 2023).Publisher: Public Library of Science Country of Publication: United States NLM ID: 101291488 Publication Model: eCollection Cited Medium: Internet

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Academic Journal

A combined ligand and target-based virtual screening strategy to repurpose drugs as putrescine uptake inhibitors with trypanocidal activity.

  • Authors : Llanos MA; Departamento de Ciencias Biológicas and Laboratorio de Investigación y Desarrollo de Bioactivos (LIDeB), Facultad de Ciencias Exactas, Universidad Nacional de La Plata. La Plata (B1900ADU), Buenos Aires, Argentina.; Alberca LN

Subjects: Trypanosoma cruzi* ; Chagas Disease*/Chagas Disease*/Chagas Disease*/drug therapy ; Chagas Disease*/Chagas Disease*/Chagas Disease*/parasitology

  • Source: Journal of computer-aided molecular design [J Comput Aided Mol Des] 2023 Feb; Vol. 37 (2), pp. 75-90. Date of Electronic Publication: 2022 Dec 10.Publisher: Springer Country of Publication: Netherlands NLM ID: 8710425 Publication Model: Print-Electronic Cited Medium: Internet ISSN:

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Academic Journal

Effect of B-NIPOx in Experimental Trypanosoma cruzi Infection in Mice.

  • Authors : Reséndiz-Mora A; Laboratorio de Biomembranas, Departamento de Bioquímica, Escuela Nacional de Ciencias Biológicas, Instituto Politécnico Nacional, Mexico City 11340, Mexico.; Laboratorio de Enzimología, Departamento de Bioquímica, Escuela Nacional de Ciencias Biológicas, Instituto Politécnico Nacional, Mexico City 11340, Mexico.

Subjects: Trypanocidal Agents*/Trypanocidal Agents*/Trypanocidal Agents*/pharmacology ; Trypanocidal Agents*/Trypanocidal Agents*/Trypanocidal Agents*/therapeutic use ; Chagas Disease*/Chagas Disease*/Chagas Disease*/drug therapy

  • Source: International journal of molecular sciences [Int J Mol Sci] 2022 Dec 25; Vol. 24 (1). Date of Electronic Publication: 2022 Dec 25.Publisher: MDPI Country of Publication: Switzerland NLM ID: 101092791 Publication Model: Electronic Cited Medium: Internet ISSN: 1422-0067

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Academic Journal

Long-term cardiology outcomes in children after early treatment for Chagas disease, an observational study.

  • Authors : González NL; Servicio de Parasitología y Chagas, Hospital de Niños Ricardo Gutiérrez, Buenos Aires, Argentina.; Moscatelli G

Subjects: Trypanocidal Agents*/Trypanocidal Agents*/Trypanocidal Agents*/therapeutic use ; Chagas Disease*/Chagas Disease*/Chagas Disease*/parasitology ; Nitroimidazoles*/Nitroimidazoles*/Nitroimidazoles*/therapeutic use

  • Source: PLoS neglected tropical diseases [PLoS Negl Trop Dis] 2022 Dec 19; Vol. 16 (12), pp. e0010968. Date of Electronic Publication: 2022 Dec 19 (Print Publication: 2022).Publisher: Public Library of Science Country of Publication: United States NLM ID: 101291488 Publication Model: eCollection Cited Medium: Internet

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Academic Journal

In Vitro and In Silico Analysis of New n-Butyl and Isobutyl Quinoxaline-7-carboxylate 1,4-di- N -oxide Derivatives against Trypanosoma cruzi as Trypanothione Reductase Inhibitors.

Subjects: Trypanosoma cruzi* ; Trypanocidal Agents*/Trypanocidal Agents*/Trypanocidal Agents*/pharmacology ; Trypanocidal Agents*/Trypanocidal Agents*/Trypanocidal Agents*/chemistry

  • Source: International journal of molecular sciences [Int J Mol Sci] 2022 Nov 01; Vol. 23 (21). Date of Electronic Publication: 2022 Nov 01.Publisher: MDPI Country of Publication: Switzerland NLM ID: 101092791 Publication Model: Electronic Cited Medium: Internet ISSN: 1422-0067

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Academic Journal

One-Pot Multicomponent Synthesis of Methoxybenzo[ h ]quinoline-3-carbonitrile Derivatives; Anti-Chagas, X-ray, and In Silico ADME/Tox Profiling Studies.

  • Authors : Ramírez H; Laboratorio de Síntesis Orgánica, Facultad de Farmacia, Universidad Central de Venezuela, Apartado 47206, Los Chaguaramos, Caracas 1041-A, Venezuela.; Facultad de Medicina, Universidad de Las Américas, Quito 170503, Ecuador.

Subjects: Chagas Disease* ; Computer Simulation* ; Quinolines*/Quinolines*/Quinolines*/chemical synthesis

  • Source: Molecules (Basel, Switzerland) [Molecules] 2021 Nov 19; Vol. 26 (22). Date of Electronic Publication: 2021 Nov 19.Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049

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Academic Journal

Vaccine-linked chemotherapy induces IL-17 production and reduces cardiac pathology during acute Trypanosoma cruzi infection.

  • Authors : Cruz-Chan JV; Texas Children's Hospital Center for Vaccine Development, Department of Pediatrics, Baylor College of Medicine, Houston, TX, USA.; Laboratorio de Parasitología, Centro de Investigaciones Regionales 'Dr. Hideyo Noguchi', Universidad Autónoma de Yucatán, Mérida, Mexico.

Subjects: Chagas Disease/Chagas Disease/Chagas Disease/*drug therapy ; Interleukin-17/Interleukin-17/Interleukin-17/*immunology ; Nitroimidazoles/Nitroimidazoles/Nitroimidazoles/*therapeutic use

  • Source: Scientific reports [Sci Rep] 2021 Feb 05; Vol. 11 (1), pp. 3222. Date of Electronic Publication: 2021 Feb 05.Publisher: Nature Publishing Group Country of Publication: England NLM ID: 101563288 Publication Model: Electronic Cited Medium: Internet ISSN:

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