Search Results

Contribution to the synthesis of positive allosteric modulators of AMPA receptors for potential use in the early diagnosis of neurodegenerative diseases.

• Authors : Lesenfants, Cindy; Goffin, Eric; Pirotte, Bernard ...

Subjects: AMPA receptors; Alzeimer's disease; AMPA positive allosteric modulators

• Source: CIRM Day, Liège, Belgium [BE], 2 février 2022

Record details

The positive allosteric modulator BPAM344 GluK2

• Authors : Bay, Yasmin; Egeberg Jeppesen, Mie; Frydenvang, Karla ...

Subjects: Cell Biology; Genetics; Molecular Biology

• Source: FEBS Letters ; volume 598, issue 7, page 743-757 ; ISSN 0014-5793 1873-3468

Record details

Exploring thienothiadiazine dioxides as isosteric analogues of benzo-and pyridothiadiazine dioxides in the search of new AMPA and kainate receptor positive allosteric modulators

• Authors : Francotte, Pierre; Bay, Yasmin; Goffin, Eric

Subjects: Ionotropic glutamate receptors Positive allosteric modulators thieno[3; 2-e]-1; 2

• Source: European Journal of Medicinal Chemistry, 264, 116036 (2023-12-09)

Record details

Total synthesis approach: development of new antimalarial compounds.

• Authors : Degotte, Gilles; Pirotte, Bernard; Frederich, Michel ...

Subjects: Malaria; Synthesis; Ellagic acidinternational

Record details

Pharmacomodulation of ellagic acid: a total synthesis approach.

• Authors : Degotte, Gilles; Pirotte, Bernard; Frederich, Michel ...

Subjects: Malaria; Ellagic acid; Pharmacomodulationinternational

Record details

Targeting Myeloperoxidase Activity and Neutrophil ROS Production to Modulate Redox Process: Effect of Ellagic Acid and Analogues.

• Authors : Degotte, Gilles; Frederich, Michel; Francotte, Pierre

Subjects: PMNs; ellagic acid; horseradish peroxidase

• Source: Molecules, 28 (11), 4516 (2023-06-02)

Record details

Design of new antimalarials inspired by ellagic acid through a total synthesis approach.

• Authors : Degotte, Gilles; Halleux, Annabelle; Pirotte, Bernard ...

Subjects: Ellagic acid; Plasmodium; Medicinal Chemistryinternational

Record details

Antiplasmodial activity of polyphenolic derivatives.

• Authors : Degotte, Gilles; Alson, Sylvain; Hans, Aurore ...

Subjects: Caffeic acid; Plasmodium; Human health sciences :: Pharmacy, pharmacology & toxicology

• Source: Antiplasmodial activity of polyphenolic derivatives. Pharmaceuticals., SwitzerlandMultidisciplinary Digital Publishing Institute (MDPI). (2019).

Record details

Preparation of ellagic acid derivatives through a total synthesis approach to improve bioavailability.

• Authors : Degotte, Gilles; Halleux, Annabelle; Hans, Aurore ...

Subjects: Ellagic acid; Plasmodium; Pharmacomodulationnational

Record details

Pharmacomodulation of ellagic acid, a promising antiplasmodial agent, to improve its bioavailability.

• Authors : Degotte, Gilles; Francotte, Pierre; Frederich, Michel ...

Subjects: Ellagic acid; Malaria; Pharmacomodulationinternational

Record details